Compound |
Property |
Calcium Assay |
IP-One Assay |
Tropicamide |
MAR anta. (M4) |
2.00 |
3.16 |
Atropine methyl bromide |
MAR anta. |
0.01 |
0.003 |
Atropine sulfate |
MAR anta. |
0.01 |
0.001 |
Atropine methyl nitrate |
MAR anta. |
0.013 |
0.001 |
BW 284c51 |
Ach. Inh. |
6.31 |
12.6 |
Aminobenztropine |
MAR anta. |
0.016 |
0.003 |
Benztropine mesylate |
MAR anta. |
0.008 |
0.013 |
4-DAMP methiodide |
M3 and M5 MAR anta. |
0.016 |
0.006 |
Dicyclomine hydrochloride |
MAR anta. |
0.039 |
0.631 |
4-DAMP mustard hydrochloride |
Irreversible MAR anta. |
0.10 |
0.126 |
L-Hyoscyamine |
MAR anta. |
0.01 |
0.501 |
Ipratropium bromide |
MAR anta. |
0.016 |
0.004 |
DL-Homatropine hydrobromide |
MAR anta. |
0.16 |
0.001 |
Hexahydro-sila-difenidol hydrochloride, p-fluoro analog |
MAR anta. |
0.16 |
1.58 |
MG 624 |
NAR anta. |
0.13 |
0.398 |
Methoctramine tetrahydrochloride |
MAR anta.(M2 selective) |
1.00 |
3.98 |
Orphenadrine hydrochloride |
MAR anta. |
0.50 |
1.00 |
Pancuronium bromide |
skeletal muscle relaxant |
10.0 |
12.6 |
Oxybutynin Chloride |
MAR anta. |
0.025 |
0.039 |
Pirenzepine dihydrochloride |
MAR anta. |
0.10 |
0.126 |
Propantheline bromide |
MAR anta. |
0.012 |
0.001 |
(-)-Scopolamine hydrobromide |
MAR anta. |
0.012 |
0.004 |
(-)-Scopolamine methyl nitrate |
MAR anta. |
0.012 |
0.001 |
(-)-Scopolamine,n-Butyl-, bromide |
MAR anta. |
0.16 |
0.50 |
(-)-Scopolamine methyl bromide |
MAR anta. |
0.013 |
0.001 |
Trihexyphenidyl hydrochloride |
MAR anta. |
0.025 |
0.0251 |
N,N,N-trimethyl-1-(4-trans-stilbenoxy)-2-propylammonium |
NAR anta. |
3.98 |
7.94 |
Telenzepine dihydrochloride |
MAR anta. (M1 select) |
0.032 |
0.025 |
WB 64 |
MAR anta. |
0.398 |
0.398 |
9-Amino-1,2,3,4-tetrahydroacridine |
Ach inh. |
15.8 |
10.0 |