Agonists | Potency, µM (Re-Screen) | Efficacy, % (Re-Screen) |
---|---|---|
retinoic acid | 0.8 | 22.2 |
CGP-7930 | 2.7 (2.6) | 18.2 (18.0) |
CGP-13501 | 2.8 (2.3) | 16.8 (15.0) |
13-cis-retinoic acid | 6.4 (2.9) | 18.8 (15.5) |
SKF-89145 hydrobromide | 21.9 (20.6) | 10.9 (16.5) |
4-hydroxybenzhydrazide | 24.6 (26.0) | 11.5 (17.5) |
Antagonists | ||
Tranilast | 0.7 (0.8) | -86 (-81.8) |
SB 205384 | 2.6 (2.5) | -75 (-73.0) |
NS-1619 | 5.2 (13.4) | -58 (-75.7) |
5-fluorouracil | 5.2 (3.1) | -72 (-71.1) |