S. No. | Comps. Code | MW |
donar HB |
accptHB | Volume | PSA |
QlogP o/w Predicted |
metab |
QPlog Khsa |
% Human Oral absorption | Violations of Rule of Five |
---|---|---|---|---|---|---|---|---|---|---|---|
1. | 355682- ASINEX |
440.50 | 3 | 5.25 | 1310.31 | 111.49 | 4.011 | 8 | 0.720 | 88.859 | 0 |
2. | 473917- ASINEX |
393.53 | 2 | 4.75 | 1293.23 | 73.29 | 4.052 | 9 | 0.853 | 92.347 | 0 |
3. | 494978- ASINEX | 398.46 | 1 | 4.5 | 1263.14 | 97.46 | 4.735 | 5 | 0.956 | 100 | 0 |
4. | 461257- ASINEX |
352.41 | 1 | 5.5 | 1152.92 | 58.58 | 3.526 | 6 | 0.497 | 92.912 | 0 |
5. | 659686-NCI | 560.64 | 2 | 11.5 | 1642.68 | 144.22 | 3.84 | 2 | 0.327 | 73.49 | 1 |
6. | 632113-NCI | 474.66 | 2 | 3.5 | 1593.61 | 62.50 | 7.472 | 3 | 1.591 | 100 | 1 |
7. | 235809-ASINEX | 502.61 | 1 | 7.5 | 1538.98 | 98.30 | 5.536 | 3 | 1.056 | 82.269 | 2 |