S. No. |
Class |
Drug |
Company |
Year of Approval |
Remarks |
Brand Name |
Active Ingredient |
1 |
NRTI |
Retrovir |
Zidovudine (AZT) |
GSK |
1987 |
|
2 |
NRTI |
Epivir |
Lamivudine (3TC) |
GSK |
1995 |
|
3 |
NRTI |
Zerit |
Stavudine (d4T) |
BMS |
1994 |
|
4 |
NRTI |
Videx |
Didanosine (ddl) |
BMS |
1989 |
|
5 |
NRTI |
Videx EC |
enteric coated didanosine (ddI EC) |
BMS |
2000 |
|
6 |
NRTI |
Ziagen |
Abacavir (ABC) |
GSK |
1988 |
|
7 |
NRTI |
Viread |
Tenovofir Disoproxil Fumarate (TDF) |
Gilead |
2002 |
|
8 |
NRTI |
Emtriva |
Emtricitabine (FTC) |
Gilead |
2003 |
|
9 |
NRTI |
Trizivir |
abacavir, zidovudine, and lamivudine (ABC, AZT and 3TC) |
GSK |
2000 |
3NRTI |
10 |
NRTI |
Combivir |
lamivudine and zidovudine (3TC and AZT) |
GSK |
1997 |
2 NRTI |
11 |
NRTI |
Epzicom |
abacavir and lamivudine (ABC and 3TC) |
GSK |
2004 |
2 NRTI |
12 |
NRTI |
Truvada |
tenofovir disoproxil fumarate and emtricitabine (TDF and FTC) |
Gilead |
2004 |
2 NRTI |
13 |
NNRTI |
Viramune |
Nevirapine (NVP) |
BI |
1996 |
|
14 |
NNRTI |
Sustiva |
Efavirenz (EFV) |
BMS |
1998 |
|
15 |
NNRTI |
Rescriptor |
Delavirdine (DLV) |
Agouron |
2003 |
|
16 |
NNRTI |
Intelence |
Etravirine |
Tibotec |
2008 |
|
17 |
NNRTI+NRTI |
Atripla |
efavirenz, emtricitabine and tenofovir disoproxil fumarate (EFV, FTC and TDF) |
Gilead |
2006 |
NNRTI+NRTI combination |
18 |
PI |
Crixivan |
Indinavir (IDV) |
Merck |
1996 |
|
19 |
PI |
Viracept |
Nelfinavir (NFV) |
Agouron |
1997 |
|
20 |
PI |
Invirase |
Saquinavir (SQV) |
Roche |
1997 |
Withdrawn 2005 |
21 |
PI |
Norvir |
Ritonavir (RTV) |
Abbott |
2000 |
|
22 |
PI |
Agenerase |
Amprenavir (APV) |
GSK |
1997 |
Withdrawn 2007 |
23 |
PI |
- |
Lopinavir (LPV) |
- |
2000 |
|
24 |
PI |
Kaletra |
Lopinavir (LPV)+Ritonavir (RTV) |
Abbott |
2005 |
2 PI |
25 |
PI |
Reyataz |
Atazanavir (ATV) |
BMS |
2003 |
|
26 |
PI |
Lexiva |
Foseamprenavir |
GSK |
2003 |
|
27 |
PI |
Prezista |
Darunvir ethanolate |
Tibotec |
2006 |
|
28 |
PI |
Aptivus |
Tipranavir (TPV) |
BI |
2005 |
|
29 |
Fusion Inhibitor |
Fuzeon |
Enfuvirtide (T-20) |
Roche |
2003 |
|
30 |
Entry Inhibitors-CCR5 co-receptor antagonist |
Selzentry |
Maraviroc |
Pfizer |
2007 |
|
31 |
HIV integrase strand transfer inhibitors |
Isentress |
Raltegravir Potassium |
Merck |
2007 |
|