Table 1:
Inhibitory Activity of the Retro -D-Sequence of DArg-D-Phe Peptides - Modified on the α-Amino Group of Arginine
№
Compounds
IC
50
µM
Ki µM
1
Cbz-D-Arg-D-Phe-OMe
110
42± 5
2
Chrom-D-Arg-D-Phe-OMe
*
56
14,35
± 0,92
3
Laur-D-Arg-D-Phe-OMe
-//-
1,76
± 0,09
*
Inhibitory effect was studied in the same buffer containing 3% DMSO in final concentration.