CB1 Analogues | EC50 (µM) | Emax (%) |
---|---|---|
A | 0.48 ± 0.03 | 112 ± 4.8 |
B | 0.22 ± 0.07 | 121 ± 1.5 |
C | 0.34 ± 0.08 | 133 ± 3.5 |
D | 0.52 ± 0.05 | 108 ± 2.7 |
E | 0.42 ± 0.03 | 103 ± 1.9 |
F | 0.27 ± 0.04 | 127 ± 4.5 |
WIN 55,212-2 | 0.18 ± 0.09 | 144 ± 6.5 |
CP-55,940 | 0.10 ± 0.05 | 135 ± 9.0 |