RECEPTORS | LIGANDS | ACTIVITY ON THE SENSORY PRIMARY NEURON |
---|---|---|
5-HT1-D | SEROTONIN | DECREASED RELEASE OF CGRP AND SUBSTANCE P |
GABA-A | GABA | DECREASED RELEASE OF CGRP AND SUBSTANCE P |
CB-1 | ANANDAMIDE* | DECREASED RELEASE OF CGRP AND SUBSTANCE P |
VR-1 | CAPSAICIN OR ANANDAMIDE** | INCREASED RELEASE OF CGRP AND SUBSTANCE P |
PAR-2 | PEPTIDIC CHAINS SLIGRL AND SLIGKV | INCREASED RELEASE OF CGRP AND SUBSTANCE P |